Description

Drug Classification:

Bisoprolol Fumarate belongs to the class of medications known as beta-blockers. Beta-blockers work by blocking the action of certain natural substances in the body, such as adrenaline, thereby reducing the workload on the heart and helping it to beat more regularly. This results in decreased blood pressure and improved heart function.

Formulations:

• Bisoprolol Fumarate Tablets:
  • Strengths: Available in 5mg and 10mg formulations.
  • Product Form: Oral tablets for convenient administration.
  • Packing Specifications: Packaged in blister packs containing 20 tablets each.

Indications:

Bisoprolol Fumarate Tablets are indicated for:

• Treatment of hypertension (high blood pressure) to lower blood pressure and reduce the risk of cardiovascular events such as heart attacks and strokes.
• Management of angina pectoris (chest pain) caused by coronary artery disease.
• Prevention of further heart failure and reduction of hospitalizations in patients with heart failure.

Usage:

• Bisoprolol Fumarate Tablets should be taken orally once daily with or without food, as directed by a healthcare professional.
• It is essential to adhere to the prescribed dosage and administration regimen to achieve optimal therapeutic outcomes.

Dosage:

• The recommended starting dose of Bisoprolol Fumarate depends on the individual patient’s condition and response to treatment.
• The usual maintenance dose ranges from 5mg to 10mg once daily, with dosage adjustment based on blood pressure and heart rate control.

Pharmacokinetics:

• Bisoprolol Fumarate is well absorbed after oral administration, with peak plasma concentrations reached within 1 to 4 hours. It undergoes hepatic metabolism and has a half-life of approximately 10 to 12 hours.
• The drug is primarily excreted in the urine as metabolites, with minimal unchanged drug excreted in the feces.

Pharmacodynamics:

• Bisoprolol Fumarate exerts its therapeutic effects by selectively blocking beta-1 adrenergic receptors in the heart, resulting in decreased heart rate, reduced myocardial contractility, and lowered blood pressure.
• By reducing the workload on the heart and decreasing oxygen demand, Bisoprolol Fumarate helps to improve symptoms and outcomes in patients with hypertension, angina, and heart failure.

Side Effects:

• Common side effects associated with Bisoprolol Fumarate Tablets may include fatigue, dizziness, headache, nausea, and diarrhea.
• Less common but potentially serious adverse effects such as bradycardia (slow heart rate), hypotension, and exacerbation of heart failure may occur and require medical attention.
• Patients should be monitored regularly for heart rate, blood pressure, and signs of worsening heart failure during treatment with Bisoprolol Fumarate Tablets.

Experience the benefits of Bisoprolol Fumarate for effective management of cardiovascular conditions, exclusively from AIT Pharmaceuticals Division. For more information, please contact us. Your heart health is our priority, and we are dedicated to providing innovative solutions for better patient care.