Description

Drug Classification:

Levocetirizine belongs to the second-generation antihistamine class of drugs. It is the active enantiomer of cetirizine, exhibiting potent antihistaminic properties with minimal sedation.

Formulations:

• Levocetirizine Tablets:
  • Strength: Each tablet contains Levocetirizine 5mg.
  • Product Form: Oral tablets for convenient administration.
  • Packing Specifications: Packaged in blister packs containing 10 tablets each.

Indications:

Levocetirizine Tablets are indicated for the relief of symptoms associated with allergic rhinitis (hay fever) and chronic idiopathic urticaria (hives). These symptoms may include sneezing, runny or itchy nose, itchy or watery eyes, itching, and skin rash.

Usage:

• Levocetirizine Tablets should be taken orally with water, preferably with or without food.
• The medication is typically used on a daily basis to manage allergy symptoms effectively.
• It is important to follow the instructions provided by a healthcare professional regarding the timing and frequency of dosing.

Dosage:

• The recommended dosage of Levocetirizine Tablets for adults and children over 12 years of age is 5mg once daily.
• For pediatric patients aged 6 to 12 years, the recommended dose is 2.5mg once daily.
• Dosage adjustment may be necessary in patients with renal impairment, as Levocetirizine is primarily eliminated via the kidneys.

Pharmacokinetics:

• Levocetirizine is rapidly absorbed from the gastrointestinal tract, with peak plasma concentrations achieved within 1 to 2 hours following oral administration.
• The drug undergoes minimal metabolism in the liver and is primarily eliminated unchanged in the urine.
• The elimination half-life of Levocetirizine is approximately 8 to 9 hours in adults, allowing for once-daily dosing.

Pharmacodynamics:

• Levocetirizine exerts its pharmacological effects by selectively antagonizing the H1 histamine receptors, thereby preventing the actions of histamine on target cells.
• By inhibiting histamine-mediated allergic responses, Levocetirizine effectively alleviates symptoms such as itching, sneezing, and nasal congestion.

Side Effects:

• Common side effects of Levocetirizine Tablets may include drowsiness, fatigue, dry mouth, headache, and gastrointestinal upset.
• Rare but serious side effects may include allergic reactions, including rash, itching, swelling, severe dizziness, and difficulty breathing.
• It is important to seek medical attention if any adverse reactions occur during treatment with Levocetirizine Tablets.

Experience the relief provided by AIT Pharmaceuticals Division’s Levocetirizine Tablets for allergy symptom management. For more information, please contact us. We are dedicated to providing effective pharmaceutical solutions to healthcare professionals worldwide.